Research Progress of Suzuki Reaction Catalyst in the Synthesis of Sartan API

Yunqi Man; Xiaolong Tan

doi:10.54097/ajst.v1i2.289

Authors

Yunqi Man
Xiaolong Tan

DOI:

https://doi.org/10.54097/ajst.v1i2.289

Keywords:

Suzuki coupling reaction, Catalyst, Research progress

Abstract

It is crucial in the pharmaceutical industry to study and develop a new class of nanocatalysts suitable for Suzuki coupling reactions and capable of being applied to the synthesis of sartans based pharmaceuticals, which are able to improve the synthesis efficiency of sartans based on their ability to resolve current scientific problems in the synthesis process, including the preparation and characterization of nanomaterial supported metal copper salt catalysts, the examination of the performance of metal catalysts in the synthesis of sartans based pharmaceuticals, and so on.

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References

Marck G, Villiger A, Buchecker R. Aryl Couplings with Heterogeneous Palladium Catalysts[J]. Tetrahedron Letters, 1994, 35(20):3277–3280.

Leblond C R, Andrews A T, Sun Y, et al. Activation of Aryl Chlorides for Suzuki Cross-Coupling by Ligandless, Heterogeneous Palladium[J]. Cheminform, 2010, 32(33):no-no.

Simeone J P, Sowa Jr J R. Palladium on carbon as a precatalyst for the Suzuki-Miyuara cross- coupling of aryl chlorides[J] Tetrahedron, 2007, 63(51): 12646-12654.

Kabalka G W, Pagni R M, Hair C M. Solventless Suzuki Coupling Reactions on Palladium-Doped KF/Al 2 O 3[J]. Organic Letters, 1999, 1(9):1423-1425.

Villemin D, Caillot F. Microwave mediated palladium-catalysed reactions on potassium fluoride/alumina without use of solvent[J]. Tetrahedron Letters, 2001, 42(4):639-642.

Kabalka GW, Pagni R M, Wang L, et al. Microwave-assisted, solventless Suzuki coupling reactions on palladium-doped alumina[J]. Green Chemistry, 2000, 2(3):120-122.

Inoue Y, Sakamoto Y, Suzuki T, et al. Organic Thin-Film Transistors with High Electron Mobility Based on Perfluoropentacene[J]. Japanese Journal of Applied Physics, 2005, 44(6A):3663-3668.

Corma A, Garc, A H, Leyva A. Bifunctional palladium-basic zeolites as catalyst for Suzuki reaction[J]. 2002, 236(1-2):179-185.

Artok L, Bulut H. Heterogeneous Suzuki reactions catalyzed by Pd(0)–Y zeolite[J]. Tetrahedron Letters, 2004, 45(20):3881-3884.

Kim Y M, Yu S. Palladium(0)-Catalyzed Amination, Stille Coupling, and Suzuki Coupling of Electron-Deficient Aryl Fluorides[J]. Journal of the American Chemical Society, 2003.

Tao Zhang, Xiujuan Feng, Mei Yan, et al Preparation of SBA-15 Supported Palladium Catalysts and their study on catalytic Suzuki coupling reactions in supercritical carbon dioxide media [J] Journal of Molecular Science: Chinese and English, 2008, 24 (1): 5

Das S, Bhunia S, Maity T, et al. Suzuki cross-coupling reaction over Pd-Schiff-base anchored mesoporous silica catalyst[J]. Journal of Molecular Catalysis A: Chemical, 2014, 394:188-197.

Gronnow M J, White R J, Clark J H, et al. Energy Efficiency in Chemical Reactions: A Comparative Study of Different Reaction Techniques[J]. Organic Process Research & Development, 2005, 9(4):516-518.

Panpranot J, Goodwin J G, Sayari A. Synthesis and characteristics of MCM-41 supported CoRu catalysts[J]. Catalysis Today, 2002, 77(3):269-284.

Chen Z, Cui Z M, Niu F, et al. Palladium Nanoparticles in Silica Hollow Spheres with Mesoporous Walls[J]. Synfacts, 2010, 2010(12):1433-1433.